SCHEMBL27967296

SCHEMBL27967296

N#Cc1ccc(Cl)c(Br)c1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.39
MAPK14 Q16539 1/20 0.35
VCAM1 P19320 2/20 0.34
CSNK1A1 P48729 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
IDO1 P14902 1/20 0.33
KDM4E B2RXH2 2/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ABL1 P00519 1/20 0.32
KDR P35968 1/20 0.32
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
KHK P50053 1/20 0.32
SLC22A12 Q96S37 2/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30881787 0.75 TRPV4 (0.39) TRPV4VCAM1KDM4EALDH1A1MAOA
SCHEMBL29209743 0.75 TRPV4 (0.39) TRPV4VCAM1KDM4EALDH1A1MAOA
SCHEMBL28327553 0.75 TRPV4 (0.39) TRPV4VCAM1ALDH1A1AR
SCHEMBL6739076 0.75 TRPV4 (0.39) TRPV4VCAM1CSNK1A1CLK4IDO1
SCHEMBL31636812 0.75 TRPV4 (0.39) TRPV4VCAM1ALDH1A1AR
SCHEMBL2657089 0.75 TRPV4 (0.39) TRPV4KDM4EUSP2ALDH1A1MAOA
SCHEMBL28245840 0.74 TRPV4 (0.42) TRPV4VCAM1CSNK1A1CLK4IDO1
SCHEMBL30352797 0.74 KDM4E (0.43) TRPV4CSNK1A1CLK4KDM4EUSP2
SCHEMBL28597079 0.74 KDM4E (0.43) TRPV4CSNK1A1CLK4KDM4EUSP2
SCHEMBL18341359 0.71 HTT (0.36) TRPV4KDM4EUSP2ALDH1A1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103842341-A Novel estrogen receptor ligands KAROBIO AB 2014-06-04 CN disclosed