SCHEMBL27970746

SCHEMBL27970746

NC1=Cc2ccccc2C1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.38
EDNRB P24530 1/20 0.38
CYP2C9 P11712 1/20 0.36
ATM Q13315 1/20 0.35
GRM1 Q13255 2/20 0.35
GRM2 Q14416 1/20 0.35
GRM4 Q14833 1/20 0.35
LMNA P02545 3/20 0.34
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 2/20 0.33
USP2 O75604 1/20 0.33
GLA P06280 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPT P10636 1/20 0.33
HDAC4 P56524 1/20 0.33
HPGD P15428 1/20 0.33
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2404932 0.81 EDNRA (0.40) EDNRAEDNRBATMGRM1GRM2
SCHEMBL2400874 0.77 EDNRA (0.37) EDNRAEDNRBCYP2C9ATMLMNA
SCHEMBL30522434 0.77 EDNRA (0.37) EDNRAEDNRBATMLMNAALDH1A1
SCHEMBL2405982 0.77 MAPT (0.44) EDNRAEDNRBCYP2C9LMNAALDH1A1
SCHEMBL8797292 0.75 HTR2A (0.43) EDNRAEDNRBCYP2C9ATMLMNA
SCHEMBL15104959 0.74 EDNRA (0.36) EDNRAEDNRBCYP2C9LMNAALDH1A1
SCHEMBL27925789 0.73 EDNRA (0.35) EDNRAEDNRBCYP2C9ATMLMNA
SCHEMBL29508252 0.73 TSHR (0.36) EDNRAEDNRBLMNAALDH1A1HDAC4
SCHEMBL5404798 0.72 EDNRA (0.34) EDNRAEDNRBLMNAALDH1A1MEN1
SCHEMBL31213694 0.72 EDNRA (0.34) EDNRAEDNRBLMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104072486-A BI-1H-BENZIMIDAZOLES AS HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO 2014-10-01 CN disclosed
CN-102177141-B bis-1H-benzimidazoles as hepatitis C virus inhibitors BRISTOL MYERS SQUIBB CO 2014-07-23 CN disclosed