SCHEMBL27971027

SCHEMBL27971027

O=[N+]([O-])c1ccc(CNc2ccc3ncsc3c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPRF P10586 1/20 0.51
PTPN2 P17706 1/20 0.51
PTPN1 P18031 1/20 0.51
PTPN11 Q06124 1/20 0.51
PRMT3 O60678 1/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KDR P35968 1/20 0.47
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28086787 0.87 MAPT (0.55) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL27980421 0.80 POLB (0.50) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL11936086 0.80 KDR (0.48) PTPN1PTPN11MEN1KMT2AKDM4E
SCHEMBL24904477 0.80 KDR (0.62) PTPN1PTPN11MEN1KMT2AKDM4E
SCHEMBL15850552 0.79 ALDH1A1 (0.51) PRMT3MAPTMEN1KMT2AALDH1A1
SCHEMBL212553 0.79 NPC1 (0.61) MEN1KMT2AKDM4EALDH1A1KDR
SCHEMBL393608 0.78 ALDH1A1 (0.53) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL11890646 0.78 MAPT (0.60) PTPN2PTPN1MAPTMEN1KMT2A
SCHEMBL11942246 0.77 KDR (0.43) PTPN1PTPN11MAPTMEN1KMT2A
Ammonia Solution, Strong SCHEMBL9639241 0.76 ALDH1A1 (0.51) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992310-B One group replaces benzo heterocyclic amine derivant and preparation method thereof and the related application as IMPDH inhibitor 中国医学科学院医药生物技术研究所 2016-07-06 CN disclosed
CN-103992310-A Group of substituted benzoheterocycle amine derivatives and preparation method and related application thereof as IMPDH (inosine monophosphate dehydrogenase) inhibitor INST MEDICINAL BIOTECHNOLOGY 2014-08-20 CN disclosed