SCHEMBL27990100

SCHEMBL27990100

Cc1c(Oc2ccc(Cl)cc2)c2cc(C[SH](=O)=O)ccc2n1CC(=O)O

nearest known ligand 0.73

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 17/20 0.73
AKR1B1 P15121 4/20 0.50
CYP2C9 P11712 2/20 0.46
MEN1 O00255 1/20 0.46
RGS12 O14924 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
PKM P14618 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
GNAI1 P63096 1/20 0.46
PMP22 Q01453 1/20 0.46
KMT2A Q03164 1/20 0.46
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049959 0.85 PTGDR2 (1.00) PTGDR2AKR1B1CYP2C9
SCHEMBL27990107 0.84 PTGDR2 (0.70) PTGDR2AKR1B1CYP2C9
SCHEMBL3372721 0.83 PTGDR2 (0.79) PTGDR2AKR1B1CYP2C9MEN1RGS12
SCHEMBL3373574 0.81 PTGDR2 (0.76) PTGDR2AKR1B1CYP2C9
SCHEMBL3372368 0.81 PTGDR2 (0.76) PTGDR2AKR1B1CYP2C9
SCHEMBL3371449 0.80 PTGDR2 (0.78) PTGDR2AKR1B1CYP2C9MEN1RGS12
SCHEMBL3371546 0.80 PTGDR2 (0.74) PTGDR2AKR1B1CYP2C9
SCHEMBL3368177 0.80 PTGDR2 (1.00) PTGDR2AKR1B1CYP2C9
SCHEMBL3372483 0.80 PTGDR2 (0.70) PTGDR2AKR1B1CYP2C9
SCHEMBL3405996 0.79 PTGDR2 (0.73) PTGDR2AKR1B1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104114169-A Combination of CRTH2 antagonist and a proton pump inhibitor for the treatment of eosinophilic esophagitis ATOPIX THERAPEUTICS LTD 2014-10-22 CN disclosed