SCHEMBL27992012

SCHEMBL27992012

Cc1cc(C)n(-c2cnc(-n3cccn3)nc2N)n1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.48
ADORA3 P0DMS8 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
TDO2 P48775 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2550961 0.80 ADORA2A (0.64) ADORA2AADORA3ADORA2BADORA1
SCHEMBL20576697 0.79 ADORA2A (0.53) ADORA2AADORA3ADORA2BADORA1MAPT
SCHEMBL2545871 0.78 ADORA2A (0.64) ADORA2AADORA3ADORA2BADORA1HTT
SCHEMBL27992067 0.72 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1HTT
SCHEMBL27992037 0.71 ADORA2A (0.60) ADORA2AADORA3ADORA2BADORA1HTT
SCHEMBL28815590 0.71 LMNA (0.42) ADORA2AADORA3ADORA2BADORA1HTT
SCHEMBL30577986 0.71 ADORA2A (0.44) ADORA2AADORA1MAPTHSD17B10KDM4E
SCHEMBL27992032 0.69 ADORA2A (0.58) ADORA2AADORA3ADORA2BADORA1KDM4E
SCHEMBL28042494 0.69 LMNA (0.42) ADORA2AADORA3ADORA2BADORA1KDM4E
SCHEMBL27991806 0.68 ADORA2A (0.47) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102892761-B 4 - aminopyrimidine derivatives and their as as adenosine a2a receptor antagonists PALOBIOFARMA SL 2015-02-04 CN claimed
CN-102892761-B 4 - aminopyrimidine derivatives and their as as adenosine a2a receptor antagonists PALOBIOFARMA SL 2015-02-04 CN disclosed