SCHEMBL27997693

SCHEMBL27997693

Cc1cc(NC(=O)c2cc(CC(C)O)n(-c3ccc(F)cc3C(F)F)c2C)ccc1S(C)(=O)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 6/20 0.57
ALDH1A1 P00352 1/20 0.39
MAPT P10636 4/20 0.35
HTT P42858 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ELANE P08246 1/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP1A2 P05177 1/20 0.33
TP53 P04637 2/20 0.33
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
ENPP2 Q13822 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MAPK1 P28482 1/20 0.32
PTGES O14684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359896 1.00 NR3C2 (0.57) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2357968 0.93 NR3C2 (0.57) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2357327 0.91 NR3C2 (0.60) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2358996 0.89 NR3C2 (0.62) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2357188 0.89 NR3C2 (0.71) NR3C2MAPTELANE
SCHEMBL27997697 0.89 NR3C2 (0.71) NR3C2MAPTELANE
SCHEMBL27997474 0.88 NR3C2 (0.66) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2358756 0.88 NR3C2 (0.66) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL2357294 0.88 NR3C2 (0.67) NR3C2ALDH1A1MAPTHTTKDM4E
SCHEMBL16456899 0.86 NR3C2 (0.46) NR3C2ALDH1A1MAPTHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102177137-B 1-phenylpyrrole compounds EXELIXIS INC 2015-03-18 CN disclosed