SCHEMBL28000643

SCHEMBL28000643

Cc1c(CCBr)cccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.40
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
KCNH2 Q12809 1/20 0.39
IDO1 P14902 2/20 0.38
PIK3C2B O00750 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
SCN8A Q9UQD0 1/20 0.35
NOTUM Q6P988 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CTSS P25774 1/20 0.35
PIK3CD O00329 2/20 0.34
PIK3CA P42336 2/20 0.34
PIK3CB P42338 2/20 0.34
PIK3CG P48736 2/20 0.34
CMA1 P23946 1/20 0.34
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30513592 0.85 P2RX7 (0.41) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL724189 0.85 P2RX7 (0.41) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL18124487 0.83 AR (0.40) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL29656253 0.83 P2RX7 (0.39) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL15532671 0.81 P2RX7 (0.41) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL10124833 0.81 P2RX7 (0.39) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL4617148 0.81 SMN1; SMN2 (0.48) P2RX7CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL3126891 0.80 IDO1 (0.52) SLC6A2SLC6A4IDO1MAOB
SCHEMBL30252413 0.80 IDO1 (0.52) SLC6A2SLC6A4IDO1MAOB
Hydrochloric Acid SCHEMBL6965231 0.80 SMN1; SMN2 (0.50) P2RX7CYP2D6SLC6A2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104395310-A Bicyclic substituted uracils and their use Bayer Pharma AG 2015-03-04 CN disclosed