SCHEMBL28002004

SCHEMBL28002004

c1ccc(CCc2cnc3ccccc3n2)nc1

nearest known ligand 0.78

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 13/20 0.78
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
HRH1 P35367 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
HRH3 Q9Y5N1 2/20 0.47
HRH4 Q9H3N8 1/20 0.47
LMNA P02545 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12066225 0.88 PDE10A (1.00) PDE10AMEN1MAPTKMT2A
SCHEMBL230753 0.79 HRH1 (0.73) MAPTHRH1CYP1A2CYP2D6HRH3
SCHEMBL29485678 0.79 HRH1 (0.73) MAPTHRH1CYP1A2CYP2D6HRH3
SCHEMBL28237594 0.79 PDE10A (0.81) PDE10AMEN1MAPTKMT2ALMNA
SCHEMBL22501412 0.78 KDM4E (0.57) PDE10AHRH1CYP1A2CYP2D6HRH3
Bromide SCHEMBL28641396 0.77 HRH1 (0.70) MAPTHRH1CYP1A2CYP2D6HRH3
SCHEMBL9971272 0.77 PDE10A (0.77) PDE10AMEN1MAPTKMT2ACYP1A2
SCHEMBL7317271 0.77 PDE10A (0.77) PDE10AMEN1MAPTKMT2ACYP1A2
SCHEMBL7317281 0.77 PDE10A (0.77) PDE10AMEN1MAPTKMT2ACYP1A2
SCHEMBL8408826 0.77 PDE10A (0.77) PDE10AMEN1MAPTKMT2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104529889-B A kind of dehydration C- alkylations of heterocyclic methyl compound 温州大学 2018-09-04 CN disclosed
CN-104529889-A Dehydration C-alkylation method for heterocyclic methyl compound UNIV WENZHOU 2015-04-22 CN disclosed