Phthalazine

Phthalazine

SCHEMBL28003247

O=Cc1ccccc1F.c1ccc2cnncc2c1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.46
NFE2L2 Q16236 3/20 0.45
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
THRB P10828 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPC1 O15118 2/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
IKBKB O14920 2/20 0.40
RAF1 P04049 1/20 0.40
RPS6KB1 P23443 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29540911 0.83
SCHEMBL87096 0.83
SCHEMBL30039913 0.83
SCHEMBL20465749 0.83
Ammonia Solution, Strong SCHEMBL30950130 0.81 MEN1 (0.60) ERN1NFE2L2LMNAMEN1THRB
Hydrazine SCHEMBL28489396 0.77 MEN1 (0.55) ERN1NFE2L2LMNAMEN1THRB
Methyl Alcohol SCHEMBL27933061 0.77 ERN1 (0.59) ERN1NFE2L2LMNAMEN1THRB
SCHEMBL4729357 0.75 ERN1 (0.57) ERN1NFE2L2LMNAMEN1THRB
Dimethylamine SCHEMBL9452721 0.75 MEN1 (0.52) ERN1NFE2L2LMNAMEN1THRB
Biphenyl SCHEMBL29187632 0.75 LMNA (0.52) ERN1NFE2L2LMNAMEN1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812746-A Bruton's tyrosine kinase inhibitors HOFFMANN LA ROCHE 2015-07-29 CN disclosed