SCHEMBL2800375

SCHEMBL2800375

CN1CCN(C(=O)C(N)COCc2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CHRM1 P11229 6/20 0.54
UGCG Q16739 8/20 0.51
CYP3A4 P08684 1/20 0.50
SLC1A1 P43005 1/20 0.49
HDAC8 Q9BY41 2/20 0.47
OPRK1 P41145 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2800372 1.00 TACR1 (0.56) TACR1HSD17B10CHRM1UGCGCYP3A4
SCHEMBL2801198 0.87 MAPT (0.46) TACR1HSD17B10CHRM1UGCG
SCHEMBL2801202 0.87 MAPT (0.46) TACR1HSD17B10CHRM1UGCG
Hydrochloric Acid SCHEMBL3791647 0.86 UGCG (0.50) TACR1UGCGCYP3A4
SCHEMBL2545138 0.86 TSHR (0.57) TACR1
Hydrochloric Acid SCHEMBL3791640 0.86 UGCG (0.50) TACR1UGCGCYP3A4
SCHEMBL2032174 0.86 GRM5 (0.62) TACR1CYP3A4SLC1A1
SCHEMBL826516 0.86 GRM5 (0.62) TACR1CYP3A4SLC1A1
Hydrochloric Acid SCHEMBL2545135 0.85 TSHR (0.56) TACR1
Hydrochloric Acid SCHEMBL2545139 0.85 TSHR (0.56) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091104-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS EXELIXIS, INC. (US) 2010-08-12 WO disclosed