SCHEMBL28005149

SCHEMBL28005149

CCOC(=O)c1ncc(OC)c(C)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.44
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
GABRA3 P34903 2/20 0.44
GABRA2 P47869 2/20 0.44
GABRA6 Q16445 2/20 0.44
DPP4 P27487 3/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TSHR P16473 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27976864 0.84 CA12 (0.44) KDM4EHPGDALDH1A1TSHRSMN1; SMN2
SCHEMBL28639867 0.77 GABRA1 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL28267255 0.76 NPSR1 (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16498192 0.74 HPGD (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL27393841 0.73 CYP2C9 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9513741 0.72 CA12 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL5820404 0.72 GABRA1 (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL460319 0.72 HTT (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10465784 0.70 TSHR (0.47) DPP4KDM4EHPGDALDH1A1TSHR
SCHEMBL27950693 0.70 HCAR2 (0.41) KDM4EHPGDALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107759516-A A kind of preparation method of the dicarboxylic acid derivatives of alkyl ether substituted pyridines 2,3 沈阳化工研究院有限公司 2018-03-06 CN disclosed
CN-104447527-A Method for preparing pyridine-2,3-dicarboxylic ester compound SINOCHEM CORP 2015-03-25 CN disclosed