SCHEMBL28005336

SCHEMBL28005336

CNC(=O)c1c(-c2ccc(F)cc2)oc2ccc(-c3cc(C(=O)NC(C)(C)C)ccc3CN)cc12

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.53
CYP3A4 P08684 5/20 0.53
KCNH2 Q12809 3/20 0.52
NR1I2 O75469 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141615 0.87 CYP2C8 (0.68) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL10240306 0.85 CYP3A4 (0.52) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005662 0.84 CYP2C8 (0.60) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005412 0.84 CYP2C8 (0.73) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL10240811 0.83 CYP3A4 (0.52) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005658 0.83 CYP3A4 (0.49) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005372 0.83 CYP2C8 (0.58) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL1919864 0.82 CYP3A4 (0.52) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005409 0.81 CYP3A4 (0.49) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL28005369 0.80 CYP2C8 (0.48) CYP2C8CYP3A4KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102209717-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2015-02-18 CN disclosed