SCHEMBL28005658

SCHEMBL28005658

CNC(=O)c1c(-c2ccc(F)cc2)oc2ccc(-c3cc(C(=O)N(CO)C4CC4)ccc3CN)cc12

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.49
CYP2C8 P10632 6/20 0.49
KCNH2 Q12809 4/20 0.48
NR1I2 O75469 1/20 0.46
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1918632 0.90 CYP3A4 (0.60) CYP3A4CYP2C8KCNH2NR1I2CYP2C9
SCHEMBL28005409 0.89 CYP3A4 (0.49) CYP3A4CYP2C8KCNH2NR1I2CYP2C9
SCHEMBL28005369 0.88 CYP2C8 (0.48) CYP3A4CYP2C8KCNH2NR1I2CYP2C9
Hydrochloric Acid SCHEMBL28005373 0.87 CYP2C8 (0.47) CYP3A4CYP2C8KCNH2NR1I2CYP2C9
SCHEMBL28005336 0.83 CYP2C8 (0.53) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL28005662 0.81 CYP2C8 (0.60) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL28005412 0.79 CYP2C8 (0.73) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL10240811 0.78 CYP3A4 (0.52) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL28005372 0.78 CYP2C8 (0.58) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL1918488 0.78 CYP3A4 (0.61) CYP3A4CYP2C8KCNH2NR1I2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102209717-B Compounds for the treatment of hepatitis c BRISTOL MYERS SQUIBB CO 2015-02-18 CN disclosed