SCHEMBL28005452

SCHEMBL28005452

CC(C)c1cc(C(C)C)c(-c2ccc(C3CCCCC3)c(C3CCCCC3)c2P(=O)(O)O)c(C(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.39
PTPN5 P54829 4/20 0.34
PTPN2 P17706 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.31
EPHX2 P34913 1/20 0.31
APP P05067 1/20 0.31
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
PTGDR2 Q9Y5Y4 2/20 0.30
PTGDR Q13258 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL161475 0.80 ROCK2 (0.43) ROCK2
SCHEMBL1013646 0.79 ROCK2 (0.47) ROCK2PTPN5PTPN2RXFP1EPHX2
SCHEMBL29470914 0.79 ROCK2 (0.47) ROCK2PTPN5PTPN2RXFP1EPHX2
SCHEMBL21044754 0.79 ROCK2 (0.43) ROCK2
SCHEMBL19643363 0.77 CA1 (0.36) PTPN5PTPN2PTGDR2PTGDR
SCHEMBL28167754 0.75 ABCB1 (0.42) PTPN5PTPN2PTGDR2
SCHEMBL27679150 0.73 PTPN5 (0.44) PTPN5PTPN2NPSR1PTGDR2
SCHEMBL28213747 0.73 ROCK2 (0.45) ROCK2EPHX2APP
SCHEMBL17868244 0.72 ROCK2 (0.40) ROCK2
SCHEMBL28796938 0.72 ROCK2 (0.36) ROCK2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104478865-B For the substituted pyrimidine for the disease for treating such as cancer 勃林格殷格翰国际有限公司 2017-09-22 CN disclosed
CN-104478865-A Substituted pyrimidines for the treatment of diseases such as cancer BOEHRINGER INGELHEIM INT 2015-04-01 CN disclosed