SCHEMBL28006388

SCHEMBL28006388

O=C1C(c2c[nH]c3ccccc23)=C(c2c[nH]c3ccccc23)C(=O)N1/N=C/c1cccc([N+](=O)[O-])c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.54
NPC1 O15118 3/20 0.54
MAPT P10636 2/20 0.54
AMY1A P0DUB6 1/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 5/20 0.47
HPGD P15428 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SIRT2 Q8IXJ6 2/20 0.46
SIRT1 Q96EB6 1/20 0.46
LMNA P02545 2/20 0.45
GAA P10253 1/20 0.44
NR1H4 Q96RI1 1/20 0.43
ELANE P08246 1/20 0.43
BCL2 P10415 1/20 0.43
MAPK1 P28482 1/20 0.43
CDK4 P11802 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28006725 0.88 MEN1 (0.52) RAB9ANPC1MAPTAMY1AHTT
SCHEMBL28006438 0.83 ELANE (0.48) RAB9ANPC1MAPTHTTALDH1A1
SCHEMBL28006734 0.83 CDK4 (0.59) RAB9ANPC1MAPTKDM4EMEN1
SCHEMBL28006432 0.83 SIRT2 (0.58) MAPTSIRT2SIRT1CDK4CDK6
SCHEMBL28006730 0.82 CDK4 (0.58) MAPTKDM4ESIRT2SIRT1CDK4
SCHEMBL28006726 0.82 SIRT2 (0.50) RAB9ANPC1MAPTHTTSIRT2
SCHEMBL28006733 0.82 SIRT2 (0.53) HPGDSIRT2SIRT1CDK4CDK6
SCHEMBL28006403 0.80 CDK4 (0.60) MAPTALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL28006405 0.80 CDK4 (0.60) MAPTALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL28818035 0.76 CDK4 (0.55) RAB9ANPC1MAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104496970-A 3,4-bi(3-indole)-2,5-dione-3-pyrrolineimine compound, preparation method of compound and application of compound in anti-cancer drug UNIV HENAN NORMAL 2015-04-08 CN disclosed