SCHEMBL28006405

SCHEMBL28006405

COc1cccc(C=NN2C(=O)C(c3c[nH]c4ccccc34)=C(c3c[nH]c4ccccc34)C2=O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 8/20 0.60
CDK6 Q00534 5/20 0.60
PRKCB P05771 1/20 0.52
SIRT2 Q8IXJ6 2/20 0.50
SIRT1 Q96EB6 1/20 0.50
ALDH1A1 P00352 3/20 0.47
RECQL P46063 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CCND1 P24385 3/20 0.44
KDR P35968 3/20 0.44
PLK4 O00444 2/20 0.44
AURKA O14965 2/20 0.44
NUAK1 O60285 2/20 0.44
FLT4 P35916 2/20 0.44
FLT3 P36888 2/20 0.44
AURKB Q96GD4 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CHRM5 P08912 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28006403 1.00 CDK4 (0.60) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006733 0.85 SIRT2 (0.53) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006734 0.84 CDK4 (0.59) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006432 0.84 SIRT2 (0.58) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006726 0.83 SIRT2 (0.50) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006730 0.83 CDK4 (0.58) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006388 0.80 RAB9A (0.54) CDK4CDK6SIRT2SIRT1ALDH1A1
SCHEMBL28006737 0.79 SIRT2 (0.57) CDK4CDK6PRKCBSIRT2SIRT1
SCHEMBL28006727 0.79 ALDH1A1 (0.57) CDK4PRKCBSIRT2SIRT1ALDH1A1
SCHEMBL28006731 0.79 ALDH1A1 (0.57) CDK4PRKCBSIRT2SIRT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104496970-A 3,4-bi(3-indole)-2,5-dione-3-pyrrolineimine compound, preparation method of compound and application of compound in anti-cancer drug UNIV HENAN NORMAL 2015-04-08 CN disclosed