SCHEMBL28008405

SCHEMBL28008405

COOCc1cccc([N+](=O)[O-])c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.59
MAOB P27338 3/20 0.56
MAOA P21397 1/20 0.56
LMNA P02545 2/20 0.53
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ACHE P22303 1/20 0.50
ALOX15 P16050 1/20 0.50
CA12 O43570 1/20 0.49
PYCR1 P32322 1/20 0.49
HTR1A P08908 1/20 0.48
ADRA1D P25100 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL791926 0.86 TSHR (0.62) TSHRMAOBMAOALMNACYP1A2
SCHEMBL1767329 0.84 TSHR (0.65) TSHRMAOBMAOALMNACYP1A2
SCHEMBL3721964 0.81 TSHR (0.57) TSHRMAOBMAOALMNACYP1A2
SCHEMBL20337575 0.81 TSHR (0.61) TSHRMAOBMAOALMNAMEN1
SCHEMBL9628070 0.81 TSHR (0.66) TSHRMAOBMAOALMNAMEN1
SCHEMBL402251 0.81 IDO1 (0.62) TSHRMAOBMAOALMNAALDH1A1
SCHEMBL5717162 0.81 TSHR (0.61) TSHRMAOBMAOALMNACYP1A2
SCHEMBL4798585 0.81 TSHR (0.61) TSHRMAOBMAOALMNACYP1A2
SCHEMBL6577663 0.80 IDO1 (0.61) TSHRMAOBLMNACYP2C19ALDH1A1
SCHEMBL11214531 0.80 TSHR (0.56) TSHRMAOBMAOALMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102746316-B An m-nitroarylmethoxy camptothecin anoxic activation prodrug for antitumor drugs JINAN TRIO PHARMATECH CO LTD 2015-04-15 CN disclosed