SCHEMBL28010664

SCHEMBL28010664

NC(=O)c1cc(-c2ccc([N+](=O)[O-])cc2)cc(-c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
CYP3A4 P08684 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
LMNA P02545 1/20 0.61
GAA P10253 1/20 0.61
POLB P06746 1/20 0.53
MAPK1 P28482 1/20 0.53
MYC P01106 1/20 0.52
MAX P61244 1/20 0.52
CA1 P00915 4/20 0.51
CA2 P00918 4/20 0.51
CA12 O43570 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51
DHODH Q02127 2/20 0.50
CES1 P23141 1/20 0.50
CASP1 P29466 1/20 0.49
TDP1 Q9NUW8 1/20 0.48
ERN1 O75460 1/20 0.48
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696165 0.87 TSHR (0.88) TSHRCYP3A4SMN1; SMN2LMNAGAA
SCHEMBL3725488 0.85 TSHR (0.68) TSHRCYP3A4SMN1; SMN2LMNAGAA
Urea SCHEMBL28797638 0.82 TSHR (0.65) TSHRLMNAGAAPOLBMAPK1
SCHEMBL9321465 0.82 CA1 (0.59) TSHRLMNAGAAPOLBMAPK1
SCHEMBL28203192 0.82 SMN1; SMN2 (0.62) TSHRCYP3A4SMN1; SMN2LMNAGAA
SCHEMBL260727 0.81 TSHR (1.00) TSHRCYP3A4SMN1; SMN2LMNAGAA
Terephthalamide SCHEMBL27950892 0.81 TSHR (1.00) TSHRCYP3A4SMN1; SMN2LMNAGAA
Nitromide SCHEMBL9225099 0.80 TSHR (0.81) TSHRCYP3A4SMN1; SMN2LMNAGAA
Hydrochloric Acid SCHEMBL11203029 0.79 TSHR (0.96) TSHRCYP3A4SMN1; SMN2LMNAGAA
SCHEMBL28194982 0.79 CYP3A4 (0.57) TSHRCYP3A4SMN1; SMN2LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104650111-A Aryl urea and aryl amide substituted oxaole pyrimindine compounds as well as preparation method and application thereof UNIV CHINA PHARMA 2015-05-27 CN disclosed