SCHEMBL28012437

SCHEMBL28012437

CCC(=O)c1ccc(OC(F)(F)C(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.54
ALDH1A1 P00352 4/20 0.51
TSHR P16473 1/20 0.51
HSD17B10 Q99714 1/20 0.51
ABCB1 P08183 2/20 0.43
MAPT P10636 4/20 0.43
HTT P42858 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
RAB9A P51151 4/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.43
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC7 Q8WUI4 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC10 Q969S8 2/20 0.43
HDAC11 Q96DB2 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141283 0.84 HDAC3 (0.54) TRPV1MAPTSMN1; SMN2RAB9AKMT2A
SCHEMBL2377766 0.83 ALDH1A1 (0.51) TRPV1ALDH1A1TSHRHSD17B10MAPT
SCHEMBL28093948 0.81 SMN1; SMN2 (0.44) ALDH1A1ABCB1MAPTHTTSMN1; SMN2
SCHEMBL2714104 0.81 TRPV1 (0.57) TRPV1ALDH1A1TSHRHSD17B10MAPT
SCHEMBL27038864 0.81 CA12 (0.53) TRPV1ALDH1A1TSHRHSD17B10MAPT
SCHEMBL9607172 0.80 EPHX2 (0.52) TRPV1MAPTSMN1; SMN2RAB9AKMT2A
SCHEMBL13019728 0.79 SMN1; SMN2 (0.48) ALDH1A1HSD17B10ABCB1MAPTHTT
SCHEMBL850939 0.79 ALDH1A1 (0.77) TRPV1ALDH1A1TSHRHSD17B10MAPT
SCHEMBL9172082 0.78 TRPV1 (0.58) TRPV1ALDH1A1TSHRHSD17B10MAPT
SCHEMBL11434818 0.78 TRPV1 (0.55) TRPV1ALDH1A1TSHRHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104520296-B Pyrrolopyridinone derivatives as TTX-S blocker 拉夸里亚创药株式会社 2016-11-16 CN disclosed
CN-104520296-A Pyrrolopyridinone derivatives as TTX-S blockers RAQUALIA PHARMA INC 2015-04-15 CN disclosed