SCHEMBL28014241

SCHEMBL28014241

O=S(=O)(c1ccc(F)cc1)c1ccc2c(c1)CNCC2

nearest known ligand 0.83

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.83
HTR2B P41595 5/20 0.83
PNMT P11086 7/20 0.76
ADRA2A P08913 1/20 0.63
ADRA2B P18089 1/20 0.63
ADRA2C P18825 1/20 0.63
HTR6 P50406 5/20 0.55
MELK Q14680 1/20 0.51
MLNR O43193 1/20 0.50
CYP2D6 P10635 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5944522 0.86 PNMT (1.00) HTR2CHTR2BPNMTADRA2AADRA2B
Hydrochloric Acid SCHEMBL5944489 0.85 PNMT (0.97) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL15435386 0.82 PNMT (0.77) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL11483387 0.81 PNMT (0.71) HTR2CHTR2BPNMTADRA2AADRA2B
Hydrochloric Acid SCHEMBL11475677 0.80 PNMT (0.69) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL29741628 0.78 PNMT (0.60) HTR2CPNMTADRA2AADRA2BADRA2C
SCHEMBL420370 0.78 PNMT (0.60) HTR2CPNMTADRA2AADRA2BADRA2C
SCHEMBL2401511 0.78 PNMT (0.71) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL29941551 0.78 PNMT (1.00) HTR2CHTR2BPNMTADRA2AADRA2B
SCHEMBL1487047 0.78 PNMT (1.00) HTR2CHTR2BPNMTADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102883607-B Compounds for the treatment of cancer GTX INC 2015-07-22 CN disclosed
CN-104592205-A COMPOUNDS FOR TREATMENT OF CANCER GTX INC 2015-05-06 CN disclosed