SCHEMBL28017273

SCHEMBL28017273

Cc1cn(C)c2cc(NC(=O)O)ncc12

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 13/20 0.69
CACNA1H O95180 1/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2298543 0.84 MAP3K5 (0.61) MAP3K5CACNA1H
SCHEMBL2297030 0.82 MAP3K5 (1.00) MAP3K5
SCHEMBL2302288 0.80 MAP3K5 (0.76) MAP3K5
SCHEMBL2300491 0.78 MAP3K5 (0.48) MAP3K5
SCHEMBL25307906 0.77 MAP3K5 (0.54) MAP3K5S1PR1S1PR3JAK1TYK2
SCHEMBL16281463 0.75 MAP3K5 (0.51) MAP3K5CACNA1H
SCHEMBL2302136 0.75 MAP3K5 (0.51) MAP3K5
SCHEMBL15031277 0.73 MAP3K5 (0.45) MAP3K5
SCHEMBL3466797 0.71 NNMT (0.44)
SCHEMBL12348928 0.71 MAP3K5 (0.62) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102834393-B Apoptosis signal-regulating kinase 1 inhibitors TAKEDA PHARMACEUTICAL 2015-07-22 CN disclosed