SCHEMBL28018561

SCHEMBL28018561

CC(=O)OC(C)(C)C(C)C#N

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
DPP4 P27487 2/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28224248 0.81 DPP4 (0.35) DPP4
SCHEMBL9709360 0.79 HCAR2 (0.36) DPP4
SCHEMBL1107368 0.76 GAA (0.44) GAATSHRALDH1A1
SCHEMBL28287215 0.72 GAA (0.41) GAATSHRALDH1A1
Acetonitrile SCHEMBL28018562 0.72 GAA (0.41) GAATSHRALDH1A1CTSSCTSK
SCHEMBL10186576 0.71 HPGD (0.44) DPP4ALDH1A1CTSK
SCHEMBL9719394 0.71
Water SCHEMBL27601078 0.70
SCHEMBL28725859 0.70 GAA (0.39) GAATSHRALDH1A1
SCHEMBL28787477 0.70 GAA (0.39) GAATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703991-B Macrocyclic Inhibitors of Flaviviridae Viruses 吉利德科学公司 2018-03-23 CN disclosed
CN-104703991-A Macrocyclic inhibitors of flaviviridae viruses GILEAD SCIENCES INC 2015-06-10 CN disclosed