SCHEMBL28021807

SCHEMBL28021807

C#Cc1cccc(-c2ccccc2C(N)=O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.59
PARP1 P09874 2/20 0.47
CHEK1 O14757 1/20 0.45
AURKA O14965 1/20 0.43
RPS6KB1 P23443 1/20 0.43
PDK2 Q15119 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
PLA2G2A P14555 3/20 0.40
PLA2G10 O15496 2/20 0.40
CTSA P10619 1/20 0.40
IKBKB O14920 2/20 0.40
SIRT2 Q8IXJ6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20703692 0.84 BCAT2 (0.59) BCAT2PARP1CHEK1PDK2IKBKB
SCHEMBL10908563 0.83 BCAT2 (0.77) BCAT2PARP1CHEK1KDM4EALDH1A1
SCHEMBL16149659 0.79 BCAT2 (0.91) BCAT2PARP1CHEK1KDM4EALDH1A1
SCHEMBL28353842 0.78 BCAT2 (0.75) BCAT2PARP1CHEK1NPC1RAB9A
SCHEMBL27597079 0.78 FABP7 (0.40) CA12CA1CA2CA9CA14
SCHEMBL28117118 0.77 PTPN1 (0.36) BCAT2PDK2ALDH1A1NPC1RAB9A
SCHEMBL1456885 0.77 BCAT2 (0.67) BCAT2PARP1CHEK1KDM4EALDH1A1
SCHEMBL28096188 0.77 BCAT2 (0.67) BCAT2PARP1CHEK1PDK2NPC1
SCHEMBL1789847 0.77 BCAT2 (0.67) BCAT2PARP1CHEK1KDM4EALDH1A1
SCHEMBL28383531 0.77 PARP1 (0.49) PARP1AURKARPS6KB1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104788333-A 2-substituted-9,10-anthraquinone compounds, and preparation method and application thereof UNIV CHINA MEDICAL 2015-07-22 CN disclosed