SCHEMBL28022326

SCHEMBL28022326

Cc1ccc2ccn(F)c2c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
CYP2A6 P11509 5/20 0.44
CYP1A2 P05177 5/20 0.44
HTR7 P34969 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
FABP4 P15090 1/20 0.36
P2RX7 Q99572 1/20 0.34
PRMT5 O14744 1/20 0.34
ROCK1 Q13464 1/20 0.33
KMO O15229 1/20 0.33
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
CYP19A1 P11511 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27995207 0.83 HTR2A (0.47) HTR2AHTR2CCYP2A6CYP1A2TDP1
SCHEMBL171810 0.76 CYP2A6 (0.55) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL20614498 0.74 HTR2A (0.47) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL28027731 0.74 HTR2A (0.47) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL27987689 0.74 HTR2A (0.47) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL7501007 0.74 HTR2A (0.51) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL15241824 0.74 HTR2A (0.51) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL13204941 0.71 HTR2C (0.53) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL10193356 0.71 HTR2C (0.62) HTR2AHTR2CCYP2A6CYP1A2HTR7
SCHEMBL13183604 0.71 HTR2A (0.45) HTR2AHTR2CCYP2A6CYP1A2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102574857-B Heterocyclic compounds as jak receptor and protein tyrosine kinase inhibitors LEO PHARMA AS 2015-06-10 CN claimed
CN-107428685-A Indole derivatives as inhibitors of dengue virus replication 杨森制药公司 2017-12-01 CN disclosed
CN-102574857-B Heterocyclic compounds as jak receptor and protein tyrosine kinase inhibitors LEO PHARMA AS 2015-06-10 CN disclosed