SCHEMBL28024062

SCHEMBL28024062

CSc1cccc(Cc2ccc(C(=O)O)cc2C(=O)O)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
KDM4E B2RXH2 2/20 0.40
CYP2C9 P11712 2/20 0.39
HIF1A Q16665 1/20 0.39
ALDH1A1 P00352 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
POLB P06746 3/20 0.36
AR P10275 1/20 0.36
NPC1 O15118 1/20 0.36
HSP90AA1 P07900 1/20 0.36
RAB9A P51151 1/20 0.36
PTPN1 P18031 1/20 0.36
LMNA P02545 2/20 0.36
AKR1C3 P42330 2/20 0.35
AKR1B10 O60218 1/20 0.35
AKR1B1 P15121 1/20 0.35
AKR1C4 P17516 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28144559 0.81 TSHR (0.47) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL28144595 0.81 TSHR (0.47) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL27994450 0.81 TSHR (0.47) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL27994717 0.81 TSHR (0.47) TSHRKDM4ECYP2C9HIF1AAR
SCHEMBL28047411 0.79 CYP2C9 (0.53) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL8889938 0.75 TSHR (0.51) TSHRCYP2C9HIF1AALDH1A1POLB
SCHEMBL28110730 0.75 GABRA1 (0.50) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL28050988 0.74 TSHR (0.48) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL28857243 0.73 TSHR (0.47) TSHRKDM4ECYP2C9HIF1AALDH1A1
SCHEMBL16316852 0.73 TSHR (0.61) TSHRKDM4ECYP2C9HIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104884442-B Terazololine-one compound and application thereof 住友化学株式会社 2016-11-02 CN disclosed
CN-104884442-A Tetrazolinone compound and applications thereof SUMITOMO CHEMICAL CO 2015-09-02 CN disclosed