SCHEMBL28024191

SCHEMBL28024191

CCOc1cc2ncccc2cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.56
PDGFRA P16234 1/20 0.56
CASP6 P55212 1/20 0.54
TLR8 Q9NR97 3/20 0.54
ALDH1A1 P00352 6/20 0.46
HSD17B10 Q99714 3/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
POLB P06746 2/20 0.46
TP53 P04637 1/20 0.46
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
TSHR P16473 1/20 0.46
CASP1 P29466 1/20 0.46
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.46
MEN1 O00255 1/20 0.46
HPGD P15428 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL360006 0.83 PDGFRB (0.74) PDGFRBPDGFRACASP6TLR8ALDH1A1
Hydrochloric Acid SCHEMBL16146746 0.82 PDGFRB (0.72) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL16146299 0.81 CASP6 (0.51) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL16146822 0.80 CASP6 (0.50) PDGFRBPDGFRACASP6TLR8ALDH1A1
Hydrochloric Acid SCHEMBL16146283 0.80 CASP6 (0.50) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL1807825 0.79 TLR8 (0.59) TLR8ALDH1A1HSD17B10KDM4EMAPT
Hydrochloric Acid SCHEMBL16146276 0.79 CASP6 (0.49) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL28251532 0.79 PDGFRB (0.57) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL357325 0.79 IRAK4 (0.48) PDGFRBPDGFRACASP6TLR8ALDH1A1
SCHEMBL3343309 0.77 CASP6 (0.57) PDGFRBPDGFRACASP6TLR8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106905234-B A method of the synthesis chloro- 6- amino -7- ethoxyquinoline of linatinib intermediate 3- cyano -4- 淮海工学院 2019-04-23 CN disclosed
CN-106905234-A A kind of method for synthesizing the ethoxyquinoline of 6 amino of HKI-272 intermediate 3 cyano group, 4 chlorine 7 淮海工学院 2017-06-30 CN disclosed
CN-104774184-A Alpha-cyano-alpha, beta-unsaturated amide compound and medical application thereof UNIV CHINA PHARMA 2015-07-15 CN disclosed