SCHEMBL28024969

SCHEMBL28024969

FC(F)(F)c1ccc(-c2nc3cncnc3[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 6/20 0.49
TNKS O95271 1/20 0.48
WNT3A P56704 1/20 0.48
TNKS2 Q9H2K2 1/20 0.48
DGAT1 O75907 4/20 0.46
KCNH2 Q12809 3/20 0.46
SCN2A Q99250 2/20 0.44
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
TRPV1 Q8NER1 2/20 0.43
KIT P10721 1/20 0.43
COMT P21964 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28818932 0.83 PIK3CA (0.41) NPBWR1DGAT1KCNH2KIT
SCHEMBL984971 0.80 NPBWR1 (0.53) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL5914424 0.80 KDM4C (0.49) TNKSTNKS2SCN2AGSK3B
SCHEMBL24075230 0.79 KIT (0.45) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL24074354 0.78 NPBWR1 (0.48) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL24075058 0.78 TNKS (0.47) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL3237120 0.78 TRPV1 (0.56) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL24074361 0.77 TRPV1 (0.51) NPBWR1TNKSWNT3ATNKS2DGAT1
SCHEMBL11352702 0.77 NPC1 (0.52) NPBWR1TNKSTNKS2SCN2ACCNB2
SCHEMBL6946824 0.76 KIT (0.45) CCNB2CDK1CCNB1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104918940-A Purine inhibitors of human phosphatidylinositol 3-kinase MERCK SHARP & DOHME 2015-09-16 CN disclosed