SCHEMBL28025835

SCHEMBL28025835

O=C(C#CBr)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.50
NTSR1 P30989 1/20 0.50
GSK3B P49841 2/20 0.48
PTPN1 P18031 1/20 0.48
MAPT P10636 5/20 0.46
CES1 P23141 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
MAPK1 P28482 2/20 0.46
CYP3A4 P08684 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 4/20 0.46
CES2 O00748 2/20 0.46
TSHR P16473 2/20 0.46
DAO P14920 1/20 0.46
NAPRT Q6XQN6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5143659 0.85 HSP90AA1 (0.57) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL10455142 0.80 CES1 (0.50) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL3523522 0.78 HSP90AA1 (0.52) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL28822400 0.77 VCP (0.56) NTSR1GSK3BMAPTCES1TDP1
SCHEMBL10829674 0.76 HSP90AA1 (0.50) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL6709770 0.76 HSP90AA1 (0.50) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL2156158 0.76 VCP (0.50) HSP90AA1NTSR1GSK3BPTPN1MAPT
SCHEMBL29136517 0.75 PTPN1 (0.41) GSK3BPTPN1MAPTCES1TDP1
SCHEMBL978641 0.74 VCP (0.75) HSP90AA1NTSR1MAPTMEN1KMT2A
SCHEMBL7464184 0.74 CES1 (0.55) HSP90AA1NTSR1MAPTCES1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104744493-B 3-benzoyl-5,7-diphenyl-5H-thiazole [3,2-a] pyrimidine derivatives and application thereof 石家庄学院 2017-01-25 CN disclosed
CN-104892640-A 2-phenyl-6-benzoyl-thiazolo[3,2-b][1,2,4]-triazole derivative and application thereof UNIV SHIJIAZHUANG 2015-09-09 CN disclosed
CN-104744493-A 3-benzoyl-5,7-diphenyl-5H-thiazole [3,2-a] pyrimidine derivatives and application thereof UNIV SHIJIAZHUANG 2015-07-01 CN disclosed