Gusperimus

Gusperimus

SCHEMBL28026

N=C(N)NCCCCCCC(=O)NC(O)C(=O)NCCCCNCCCN

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 8/20 0.47
CHRNB2 P17787 3/20 0.44
CHRNB4 P30926 3/20 0.44
CHRNA3 P32297 3/20 0.44
CHRNA4 P43681 3/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRM1 Q13255 2/20 0.44
PAOX Q6QHF9 1/20 0.43
CHRNA1 P02708 1/20 0.41
CHRNG P07510 1/20 0.41
CHRNB1 P11230 1/20 0.41
CHRND Q07001 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9772173 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9772156 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9688242 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL8656104 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL25482108 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL12980163 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL26925 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL317912 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9772186 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9772231 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12914 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4745155-A1 POWDER CONTAINING PARTICLES OF GELATIN DERIVATIVE AND APPLICATION OF SAME IN MEDICAL TREATMENT National Institute for Materials Science (JP) 2026-05-20 EP claimed
US-12571044-B2 Classifier for identification of robust sepsis subtypes THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-03-10 US claimed
US-20250295638-A1 METHODS OF TREATING ALLOGRAFT REJECTION BARGENT THERAPEUTICS PTY LTD (AU) 2025-09-25 US claimed
EP-4578454-A1 COMPOSITIONS COMPRISING PLATELET DERIVED EXTRACELLULAR VESICLES Lysatpharma GmbH (DE) 2025-07-02 EP claimed
EP-4518857-A1 METHODS OF TREATING ALLOGRAFT REJECTION Bargent Therapeutics Pty Limited (AU) 2025-03-12 EP claimed
WO-2025029671-A1 CELL THERAPY FOR DIABETES VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-02-06 WO claimed
WO-2025013818-A1 POWDER CONTAINING PARTICLES OF GELATIN DERIVATIVE AND APPLICATION OF SAME IN MEDICAL TREATMENT 国立研究開発法人物質・材料研究機構 2025-01-16 WO claimed
EP-4473088-A2 CELL THERAPY FOR DIABETES Vertex Pharmaceuticals Incorporated (US) 2024-12-11 EP claimed
EP-3773563-B1 PRODRUGS OF FUSED-BICYCLIC C5AR ANTAGONISTS CHEMOCENTRYX INC (US) 2024-10-16 EP claimed
CN-118354776-A Methods and compositions for enhanced efficacy and reduced toxicity of non-implanted CD8 depleted allogeneic donor lymphocyte infusions 约翰霍普金斯大学 2024-07-16 CN claimed
WO-1995015770-A1 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1995-06-15 WO claimed
WO-1995001786-A1 PHARMACEUTICAL COMPOSITIONS FOR HARDLY SOLUBLE ACTIVE SUBSTANCES CIBA-GEIGY AG (CH) 1995-01-19 WO claimed
EP-0359347-B1 COVALENTLY-LINKED COMPLEXES AND METHODS FOR ENHANCED CYTOTOXICITY AND IMAGING NEORX CORPORATION (US) 1992-12-23 EP claimed
CN-1017621-B Process for preparing crystalline deoxyspergualin TAKARA SHIY ZOU CO LTD (JP) 1992-07-29 CN claimed
CN-1047670-A Crystalline deoxyspergualin (deoxyspergualin) and preparation method thereof TAKARA SHIY ZOU CO LTD (JP) 1990-12-12 CN claimed
EP-0400889-A1 Crystalline deoxyspergualin and process for its preparation TAKARA SHUZO CO. LTD. (JP) 1990-12-05 EP claimed
EP-0359347-A2 Covalently-linked complexes and methods for enhanced cytotoxicity and imaging NEORX CORPORATION (US) 1990-03-21 EP claimed
US-4876244-A STABILIZERS OF DEXTRANS, CYCLODEXTRINS, AND CHONDROITIN SULFATE; ANTICARCINOGENIC AGENTS, IMMUNOMODULATORS ZAIDAN HOJIN BISEIBUTSU KAGAKU (JP) 1989-10-24 US claimed
US-4710517-A MALTOSE, LACTOSE STABILIZERS; ANTICARCINOGENIC AGENTS, IMMUNOMODULATORS ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1987-12-01 US claimed
US-4518532-A ANTITIMOR ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1985-05-21 US claimed