Gusperimus

Gusperimus

SCHEMBL8656104

N=C(N)NCCCCCCC(=O)N[C@@H](O)C(=O)NCCCCNCCCN

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 8/20 0.47
CHRNB2 P17787 3/20 0.44
CHRNB4 P30926 3/20 0.44
CHRNA3 P32297 3/20 0.44
CHRNA4 P43681 3/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRM1 Q13255 2/20 0.44
PAOX Q6QHF9 1/20 0.43
CHRNA1 P02708 1/20 0.41
CHRNG P07510 1/20 0.41
CHRNB1 P11230 1/20 0.41
CHRND Q07001 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9772173 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL28026 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9772156 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9688242 1.00 GRIA1 (0.47) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL25482108 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL12980163 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL26925 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Gusperimus SCHEMBL317912 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9772186 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9772231 0.99 GRIA1 (0.46) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755380-B1 15-DEOXYSPERGUALIN ANALOGS, THERAPEUTICAL USE THEREOF, AND METHOD FOR PREPARING SAME FOURNIER IND & SANTE (FR) 1998-10-14 EP disclosed