SCHEMBL28026045

SCHEMBL28026045

CC(=O)N(C)CCN1CCC(c2ccccc2)(N2CCCC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.55
SIGMAR1 Q99720 2/20 0.48
GRIN2D O15399 1/20 0.48
GRIN3B O60391 1/20 0.48
CYP2B6 P20813 1/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
PRCP P42785 1/20 0.48
SLC6A3 Q01959 1/20 0.48
GRIN1 Q05586 1/20 0.48
KCNH2 Q12809 1/20 0.48
GRIN2A Q12879 1/20 0.48
GRIN2B Q13224 1/20 0.48
GRIN2C Q14957 1/20 0.48
GRIN3A Q8TCU5 1/20 0.48
OPRM1 P35372 2/20 0.47
OPRD1 P41143 1/20 0.47
KDM1A O60341 1/20 0.46
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2331745 0.91 HRH3 (0.56) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
Hydrochloric Acid SCHEMBL2333142 0.90 HRH3 (0.55) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL2831968 0.85 HRH3 (0.50) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL2333546 0.82 HRH3 (0.47) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL3409607 0.80 ALDH1A1 (0.46) HRH3
SCHEMBL28026517 0.79 KDM4E (0.45) HRH3
SCHEMBL3404217 0.79 HRH3 (0.44) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL3410705 0.78 HRH3 (0.43) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL3403655 0.78 HRH3 (0.43) HRH3SIGMAR1GRIN2DGRIN3BCYP2B6
SCHEMBL3409858 0.77 HSD17B10 (0.44) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102015683-B The indole derivatives replaced GRUNENTHAL GMBH (DE) 2015-08-05 CN claimed
CN-102015683-B The indole derivatives replaced GRUNENTHAL GMBH (DE) 2015-08-05 CN disclosed