SCHEMBL28026318

SCHEMBL28026318

CC(Br)c1ccc(N)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.46
NOS2 P35228 2/20 0.46
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 1/20 0.41
GABRP O00591 2/20 0.36
GABRD O14764 2/20 0.36
GABRA1 P14867 2/20 0.36
GABRB1 P18505 2/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
GABRA5 P31644 2/20 0.36
GABRA3 P34903 2/20 0.36
GABRA2 P47869 2/20 0.36
GABRB2 P47870 2/20 0.36
GABRA4 P48169 2/20 0.36
GABRE P78334 2/20 0.36
GABRA6 Q16445 2/20 0.36
GABRG1 Q8N1C3 2/20 0.36
GABRG3 Q99928 2/20 0.36
GABRQ Q9UN88 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL83975 0.82 NOS3 (0.50) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL31222667 0.82 NOS3 (0.50) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL14647750 0.80 NOS3 (0.48) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL4328494 0.80 NOS3 (0.48) NOS3NOS2KDM4EHSD17B10GABRP
Hydrochloric Acid SCHEMBL23201276 0.78 NOS3 (0.46) NOS3NOS2KDM4EHSD17B10GABRP
Hydrochloric Acid SCHEMBL30929411 0.78 NOS3 (0.46) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL27461381 0.78 NOS3 (0.46) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL23478507 0.78 NOS3 (0.46) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL6469008 0.78 NOS3 (0.46) NOS3NOS2KDM4EHSD17B10GABRP
SCHEMBL24703386 0.77 NOS3 (0.45) NOS3NOS2KDM4EHSD17B10GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104981466-A novel antibacterial compounds JANSSEN SCIENCES IRELAND UC 2015-10-14 CN disclosed
CN-104781250-A New antibacterial compounds JANSSEN SCIENCES IRELAND UC 2015-07-15 CN disclosed
CN-102656158-B Novel heterocyclic acrylamides and their use as pharmaceuticals FAB PHARMA SAS 2015-02-11 CN disclosed
CN-104119331-A Alkenyl compound as well as use method and application thereof GUANGDONG HEC PHARMACEUTICAL 2014-10-29 CN disclosed
CN-103459384-A Benzoxazepines as inhibitors of PI3K/mTOR and methods of their use and manufacture EXELIXIS INC 2013-12-18 CN disclosed