Ziprasidone

Ziprasidone

SCHEMBL28028

O=C1Cc2cc(CCN3CCN(c4nsc5ccccc45)CC3)c(Cl)cc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2HTR2AHTR2C

The experimentally established mechanism targets of Ziprasidone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 13/20 1.00
DRD2 known ✓ P14416 11/20 1.00
HTR2C known ✓ P28335 1/20 1.00
HTR1A P08908 8/20 1.00
HTR7 P34969 3/20 1.00
KCNH2 Q12809 2/20 1.00
HTR6 P50406 2/20 1.00
HTR3E A5X5Y0 1/20 1.00
HTR3B O95264 1/20 1.00
ABCB11 O95342 1/20 1.00
PGR P06401 1/20 1.00
CHRM2 P08172 1/20 1.00
ADRA2A P08913 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
MAPT P10636 1/20 1.00
CHRM1 P11229 1/20 1.00
GOT1 P17174 1/20 1.00
ADRA2B P18089 1/20 1.00
ADRA2C P18825 1/20 1.00
DRD1 P21728 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ziprasidone SCHEMBL29368426 1.00 HTR2A (1.00) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL4774002 1.00 HTR2A (1.00) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL30354044 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL3139060 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL122876 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL5859456 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL3143295 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL4914143 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL6599516 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2
Ziprasidone SCHEMBL374870 0.99 HTR2A (0.98) HTR2ADRD2HTR1AHTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 25062 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122079853-A N-substituted indoles and other heterocyclic compounds for the treatment of brain diseases 2026-05-26 CN claimed
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
WO-2026106952-A1 METHODS FOR TREATING CONGENITAL DISORDERS OF GLYCOSYLATION CDG CARE (US) 2026-05-21 WO claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-12624036-B2 Method of treating post-traumatic stress disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
US-12624037-B2 Method of treating agitation, aggressive behavior, and impulse control disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
US-12617809-B2 Cardioprotective lipid and method of use SIGNPATH PHARMA, INC. (US) 2026-05-05 US claimed
WO-2026090360-A1 FUSED PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC. (US) 2026-04-30 WO claimed
US-20260108529-A1 FUSED AMINO PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, ACUTE SENSORINEURAL HEARING LOSS, AGE-RELATED HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC (US) 2026-04-23 US claimed
WO-1997032037-A1 ASSESSMENT OF THE RESPONSIVENESS OF INDIVIDUALS TO MODULATORS OF THE 5-HT2 RECEPTORS, ESPECIALLY THE 5-HT2A RECEPTOR SMITHKLINE BEECHAM PLC (GB) 1997-09-04 WO claimed
EP-0790236-A1 Pro-drugs of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2h-indol-2-one PFIZER INC. (US) 1997-08-20 EP claimed
WO-1997021833-A1 METHOD OF PREDICTING A SUBJECTS RESPONSE TO NEUROLEPTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-19 WO claimed
CN-1142945-A Medcine for curing cerebrovascular disturbance with psychonosema SUMITOMO PHARMA (JP) 1997-02-19 CN claimed
CN-1033089-C Process for preparation aryl piperazinyl-heterocyclic compounds PFIZER (US) 1996-10-23 CN claimed
WO-1996031621-A2 METHOD FOR DETERMINING THE RESPONSIVENESS OF INDIVIDUALS TO 5-HT2 RECEPTOR MODULATING AGENTS SMITHKLINE BEECHAM PLC (GB) 1996-10-10 WO claimed
EP-0730865-A1 Use of serotonin and dopamine receptor blockers for the treatment of mental disorders associated with cerebrovascular disease SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-09-11 EP claimed
US-5338846-A Process for preparing aryl piperazinyl-heterocyclic compounds with a piperazine salt PFIZER INC. (US) 1994-08-16 US claimed
EP-0586191-A1 Monohydrate of 5-(2-(4-(1,2 Benzisothiazol-3-YL)-1-Piperazinyl)-Ethyl)-6-Chloro-1,3-Dihydro-2H-indol-2-one Hydrochloride PFIZER INC. (US) 1994-03-09 EP claimed
EP-0584903-A1 Process for preparing aryl piperazinyl-heterocyclic compounds PFIZER INC. (US) 1994-03-02 EP claimed