SCHEMBL28028147

SCHEMBL28028147

CN(C)C1CCN(c2c[c]ccn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
MAP4K4 O95819 1/20 0.36
KIT P10721 2/20 0.35
FLT3 P36888 2/20 0.35
CXCR4 P61073 1/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
PDE10A Q9Y233 2/20 0.34
OPRD1 P41143 1/20 0.34
IKBKB O14920 1/20 0.34
WNT1 P04628 2/20 0.33
GSK3B P49841 2/20 0.33
DYRK1A Q13627 2/20 0.33
PARP1 P09874 1/20 0.33
PTPN11 Q06124 1/20 0.33
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33
CDK4 P11802 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4831454 0.77 HRH4 (0.34) HRH4
SCHEMBL1599784 0.77 HRH4 (0.38) HRH4CXCR4
SCHEMBL4781342 0.76 ALDH1A1 (0.37)
SCHEMBL1569984 0.76 HRH4 (0.45) HRH4HRH3
SCHEMBL2324452 0.75 HRH4 (0.40) HRH4MAP4K4CXCR4
SCHEMBL22837819 0.75 PLD1 (0.53)
SCHEMBL933191 0.74 MAP4K4 (0.39) HRH4HRH3MAP4K4KITFLT3
SCHEMBL27549279 0.74 PDE10A (0.40) PDE10A
SCHEMBL455110 0.73 PIK3CA (0.44)
SCHEMBL182823 0.73 PLD1 (0.53) HRH4HRH3DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed