SCHEMBL28028671

SCHEMBL28028671

Nc1cccc(C2COCCN2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 1/20 0.59
PRKACG P22612 1/20 0.59
PRKACB P22694 1/20 0.59
MAP4K1 Q92918 2/20 0.39
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
CTSK P43235 1/20 0.35
CYP3A4 P08684 1/20 0.34
CASP1 P29466 1/20 0.34
RECQL P46063 1/20 0.34
ATR Q13535 1/20 0.33
CSNK1D P48730 1/20 0.33
CSNK1E P49674 1/20 0.33
KCNH2 Q12809 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1A P35348 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MAOA P21397 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22425354 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBMAP4K1CTSK
SCHEMBL7353494 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBCSNK1DCSNK1E
SCHEMBL21723230 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBCSNK1DCSNK1E
SCHEMBL28785154 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBMAP4K1CTSK
SCHEMBL14839631 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBCTSKHTR2B
SCHEMBL432870 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBMAP4K1CTSK
SCHEMBL22425356 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBMAP4K1CTSK
SCHEMBL30824548 0.81 PRKACA (0.52) PRKACAPRKACGPRKACBMAP4K1CTSK
SCHEMBL3399522 0.80 PRKACA (0.47) PRKACAPRKACGPRKACBMAP4K1DDB1
Hydrochloric Acid SCHEMBL25320856 0.79 PRKACA (0.51) PRKACAPRKACGPRKACBMAP4K1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed