SCHEMBL28030557

SCHEMBL28030557

O=[N+]([O-])c1ccc2cnc(Br)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
CYP3A4 P08684 3/20 0.46
NOS1 P29475 2/20 0.46
LMNA P02545 2/20 0.46
ALOX15 P16050 1/20 0.46
POLB P06746 1/20 0.46
MAOB P27338 1/20 0.46
ALDH1A1 P00352 5/20 0.44
TDP1 Q9NUW8 2/20 0.41
NAMPT P43490 1/20 0.40
XDH P47989 1/20 0.40
TSHR P16473 2/20 0.39
CYP1A2 P05177 1/20 0.39
GLS O94925 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TXNRD1 Q16881 1/20 0.39
TXNRD3 Q86VQ6 1/20 0.39
TXNRD2 Q9NNW7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17374976 0.93 MAPT (0.46) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL28030111 0.79 HSD17B10 (0.47) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL16307679 0.79 CYP1A2 (0.48) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL3829978 0.77 TSHR (0.56) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL14010958 0.76 MAPT (0.53) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL30095409 0.76 MAPT (0.53) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL28338203 0.75 TSHR (0.54) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL27981594 0.75 ALDH1A1 (0.46) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL28122579 0.74 TSHR (0.59) MAPTCYP3A4NOS1LMNAALOX15
SCHEMBL5778139 0.74 SNCA (0.50) MAPTCYP3A4NOS1LMNAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017152-B Preparation method of 3-chloro-6-nitroisoquinoline or 3-bromine-6-nitroisoquinoline 北京六合宁远科技有限公司 2017-05-10 CN disclosed
CN-105017152-B Preparation method of 3-chloro-6-nitroisoquinoline or 3-bromine-6-nitroisoquinoline 北京六合宁远科技有限公司 2017-05-10 CN disclosed
CN-105017152-A Preparation method of 3-chloro(bromo)-6-nitroisoquinoline BEIJING LIUHE NINGYUAN TECHNOLOGY CO LTD 2015-11-04 CN disclosed