SCHEMBL28032029

SCHEMBL28032029

Cc1c(N=[N+]=[N-])cccc1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.58
TSHR P16473 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ALDH1A1 P00352 3/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
GRIA2 P42262 1/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
GPR35 Q9HC97 1/20 0.40
PLAU P00749 1/20 0.40
GAA P10253 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356198 0.82 PLAU (0.53) TDP1TSHRALDH1A1GRIA2KMT2A
SCHEMBL16329327 0.82 PLAU (0.53) TDP1TSHRALDH1A1GRIA2KMT2A
SCHEMBL38656863 0.80 TDP1 (0.44) TDP1TSHRSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL18887676 0.79 TDP1 (0.67) TDP1TSHRSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL16774460 0.78 CYP3A4 (0.43) TSHR
SCHEMBL8222001 0.77 TDP1 (0.64) TDP1TSHRSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL3305095 0.77 TDP1 (0.64) TDP1TSHRSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL19569929 0.77 TDP1 (0.48) TDP1TSHRSMN1; SMN2ALDH1A1GRIA2
SCHEMBL13019646 0.76 TDP1 (0.62) TDP1TSHRSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL472112 0.75 TDP1 (1.00) TDP1TSHRSMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527332-B Biological activity-possessed caspovir derivative, and preparation method and application thereof 南开大学 2022-07-26 CN claimed
CN-113527333-A Dolutegravir derivative with biological activity and preparation method and application thereof 南开大学 2021-10-22 CN claimed
CN-113527332-A Kabauvir derivative with biological activity and preparation method and application thereof 南开大学 2021-10-22 CN claimed
CN-114671874-B Theophylline acetic acid derivative with anti-tumor activity and preparation method and application thereof 济南爱思医药科技有限公司 2024-02-02 CN disclosed
CN-113527333-B Dolutegravir derivative with biological activity and preparation method and application thereof 南开大学 2022-08-05 CN disclosed
CN-113527332-B Biological activity-possessed caspovir derivative, and preparation method and application thereof 南开大学 2022-07-26 CN disclosed
CN-114671874-A Theophylline acetic acid derivative with anti-tumor activity and preparation method and application thereof 济南爱思医药科技有限公司 2022-06-28 CN disclosed
CN-113980022-B Theophylline acetic acid derivative with antitumor activity and preparation method thereof 南开大学 2022-06-21 CN disclosed
CN-113980022-A Theophylline acetic acid derivative with antitumor activity and preparation method thereof 南开大学 2022-01-28 CN disclosed
CN-113527333-A Dolutegravir derivative with biological activity and preparation method and application thereof 南开大学 2021-10-22 CN disclosed
CN-113527332-A Kabauvir derivative with biological activity and preparation method and application thereof 南开大学 2021-10-22 CN disclosed
CN-104876913-B Preparation method of 4,6-dimethyl-2-thiopyrimidine-1,2,3-triazole compound with antitumor activity 河南师范大学 2017-01-25 CN disclosed
CN-104876913-A Preparation method of 4,6-dimethyl-2-thiopyrimidine-1,2,3-triazole compound with antitumor activity UNIV HENAN NORMAL 2015-09-02 CN disclosed