SCHEMBL28033848

SCHEMBL28033848

CCOC(=O)c1nc(N)ccc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
CYP1A2 P05177 3/20 0.49
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 2/20 0.48
MAPK1 P28482 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAOA P21397 1/20 0.47
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 2/20 0.44
NPC1 O15118 2/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
MPI P34949 1/20 0.43
HPGD P15428 1/20 0.43
TARBP2 Q15633 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1269540 0.83 ALDH1A1 (0.46) ALDH1A1CYP1A2KMT2AKDM4EL3MBTL1
SCHEMBL4162744 0.83 KDM4E (0.48) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
SCHEMBL29756221 0.82 NPSR1 (0.48) ALDH1A1KMT2AKDM4EL3MBTL1HSD17B10
SCHEMBL13406205 0.82 KDM4E (0.50) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
SCHEMBL267964 0.82 NPSR1 (0.48) ALDH1A1KMT2AKDM4EL3MBTL1HSD17B10
SCHEMBL8309273 0.81 KDM4E (0.49) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
SCHEMBL26172461 0.79 TARBP2 (0.48) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
SCHEMBL19609345 0.79 ALDH1A1 (0.45) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
Hydrochloric Acid SCHEMBL19583715 0.78 ALDH1A1 (0.44) ALDH1A1CYP1A2KMT2AKDM4EMAPK1
SCHEMBL1680317 0.76 ALDH1A1 (0.54) ALDH1A1CYP1A2KMT2AKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085429-A Heteroaromatic derivative and application thereof to medicament GUANGDONG HEC PHARMACEUTICAL 2015-11-25 CN disclosed