SCHEMBL28034150

SCHEMBL28034150

COc1ccc2c(O)nc(-c3ccc(C(C)C)cc3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
CASP3 P42574 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CASR P41180 1/20 0.44
ABCB11 O95342 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTGS2 P35354 3/20 0.40
AKR1C3 P42330 3/20 0.40
AKR1C2 P52895 3/20 0.40
PTGS1 P23219 2/20 0.40
CDC42 P60953 1/20 0.40
RAC1 P63000 1/20 0.40
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13728566 0.86 ACP1 (0.47) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8348782 0.86 NPC1 (0.47) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL28033683 0.85 NPC1 (0.46) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL13730043 0.83 NPC1 (0.49) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8272309 0.83 NPC1 (0.57) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8348779 0.82 PDGFRB (0.47) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL13728430 0.82 KMO (0.45) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8351874 0.81 APP (0.48) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8186120 0.80 ACP1 (0.45) NPC1RAB9ACASP3SENP7KDM4E
SCHEMBL8272618 0.78 KDM4E (0.45) NPC1RAB9ACASP3SENP7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103797024-B Hepatitis c virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2016-06-01 CN disclosed
CN-104918941-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-09-16 CN disclosed