SCHEMBL28035688

SCHEMBL28035688

COc1c[c]c(-c2c(O)cc(O)cc2O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MAPK1 P28482 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
CYP1A2 P05177 1/20 0.41
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
ALOX12 P18054 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28514922 0.81 GAA (0.43) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL1420029 0.75 ESR2 (0.59) NPC1RAB9AMAPK1SMN1; SMN2TP53
SCHEMBL8591645 0.70 CA1 (0.48) NPC1RAB9AMAPK1SMN1; SMN2TP53
SCHEMBL1029610 0.69
SCHEMBL16056542 0.67 CYP3A4 (0.48) NPC1RAB9AMAPK1SMN1; SMN2TP53
SCHEMBL6417992 0.67 CA4 (0.44) NPC1RAB9ASMN1; SMN2CYP1A2KDM4E
SCHEMBL16400853 0.67 CYP1A2 (0.41) NPC1RAB9ASMN1; SMN2CYP1A1CYP1B1
SCHEMBL27934853 0.66 CYP3A4 (0.46) NPC1RAB9AMAPK1SMN1; SMN2TP53
SCHEMBL6950427 0.66 NPC1 (0.45) NPC1RAB9AMAPK1SMN1; SMN2TP53
SCHEMBL16318731 0.65 TNIK (0.38) NPC1RAB9AMAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112321579-A Salts of 2-amino-1-hydroxyethyl-8-hydroxyquinolin-2 (1H) -one derivatives 阿尔米雷尔有限公司 2021-02-05 CN disclosed
CN-103649089-B Pyrrolotriazinones as PI3K inhibitors 阿尔米雷尔有限公司 2016-06-29 CN disclosed
CN-105492027-A Salts of 2-amino-1-hydroxyethyl-8-hydroxyquinolin-2 (1H) -one derivatives having both muscarinic receptor antagonist and beta 2 adrenergic receptor agonist activity ALMIRALL SA 2016-04-13 CN disclosed
CN-105025897-A Salts of 2-amino-1-hydroxyethyl-8-hydroxyquinolin-2 (1H) -one derivatives having both beta 2 adrenergic receptor agonist and M3 muscarinic receptor antagonist activity ALMIRALL SA 2015-11-04 CN disclosed