SCHEMBL6417992

SCHEMBL6417992

COc1c[c]c(-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA4 P22748 1/20 0.44
LTA4H P09960 2/20 0.43
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
BACE1 P56817 2/20 0.41
TRPA1 O75762 1/20 0.39
MITF O75030 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591645 0.88 CA1 (0.48) NPC1RAB9AKDM4ETDP1BACE1
SCHEMBL1420156 0.82 MAOB (0.50) NPC1RAB9AALDH1A1LMNANPSR1
SCHEMBL28208024 0.81 MEN1 (0.42) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL1420029 0.81 ESR2 (0.59) LTA4HNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL28904555 0.81 APP (0.41) NPC1RAB9ASMN1; SMN2CA12CA1
SCHEMBL28961082 0.79 LTA4H (0.48) LTA4HNPC1RAB9AKDM4EALDH1A1
SCHEMBL28150942 0.78 ESR2 (0.48) NPC1RAB9AKDM4ETDP1BACE1
SCHEMBL28433765 0.76 METAP2 (0.36) SMN1; SMN2MAPT
SCHEMBL27860514 0.76 APP (0.43) CA4ALDH1A1L3MBTL1HTTSMN1; SMN2
SCHEMBL7123909 0.73 HPGD (0.42) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116768796-A Novel pyrazole-3-carboxamide derivative and preparation method and application thereof 河北农业大学 2023-09-19 CN claimed
CN-111087338-B Sulfonamide-substituted pyrrolidones derivative and preparation method thereof 常州大学 2021-03-02 CN claimed
CN-111087338-A Sulfonamide-substituted pyrrolidones derivative and preparation method thereof 常州大学 2020-05-01 CN claimed
CN-116768796-A Novel pyrazole-3-carboxamide derivative and preparation method and application thereof 河北农业大学 2023-09-19 CN disclosed
CN-112390697-B Synthesis method of N-arylselenium/thioethyl sulfoxide imine 成都理工大学 2023-03-10 CN disclosed
CN-107353233-B Method for catalytic synthesis of asymmetric azoxybenzene compound 温州大学 2023-02-24 CN disclosed
CN-111087338-B Sulfonamide-substituted pyrrolidones derivative and preparation method thereof 常州大学 2021-03-02 CN disclosed
CN-112390697-A Synthesis method of N-arylselenium/thioethyl sulfoxide imine 成都理工大学 2021-02-23 CN disclosed
CN-108424377-B Method for synthesizing asymmetric azoxybenzene compound 温州大学 2021-02-19 CN disclosed
CN-108689890-B Method for synthesizing asymmetric azoxybenzene compound 温州大学 2020-11-17 CN disclosed
CN-111087338-A Sulfonamide-substituted pyrrolidones derivative and preparation method thereof 常州大学 2020-05-01 CN disclosed
CN-108689890-A A kind of synthetic method of asymmetric azobenzene oxide compound 温州大学 2018-10-23 CN disclosed
CN-108424377-A A kind of synthetic method of asymmetric oxidation azobenzene compound 温州大学 2018-08-21 CN disclosed
CN-107353233-A A kind of method for catalyzing and synthesizing asymmetric oxidation azobenzene compound 温州大学 2017-11-17 CN disclosed
WO-2005092896-A1 COMPOUND FOR INHIBITING TYROSINE KINASE ACTIVITY OF DDR2 PROTEIN KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2005-10-06 WO disclosed