SCHEMBL28035907

SCHEMBL28035907

CCCCn1nc(-c2ccc(F)cc2)cc1C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 13/20 0.50
HDAC3 O15379 11/20 0.50
HDAC4 P56524 11/20 0.50
HDAC1 Q13547 11/20 0.50
HDAC2 Q92769 11/20 0.50
HDAC8 Q9BY41 11/20 0.50
HDAC7 Q8WUI4 10/20 0.50
HDAC10 Q969S8 10/20 0.50
HDAC11 Q96DB2 10/20 0.50
HDAC9 Q9UKV0 10/20 0.50
HDAC5 Q9UQL6 10/20 0.50
SMPD1 P17405 1/20 0.46
NCOR2 Q9Y618 3/20 0.43
TLR8 Q9NR97 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TGFBR1 P36897 1/20 0.41
TGFBR2 P37173 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28014600 0.87 HDAC6 (0.59) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL5333233 0.79 HDAC3 (0.55) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28035847 0.77 SMPD1 (0.67) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL11393727 0.76 HSD17B10 (0.50) KDM4EALDH1A1
SCHEMBL25229993 0.75 SMN1; SMN2 (0.57) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28013853 0.74 HDAC6 (0.60) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28013855 0.73 HDAC6 (0.59) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL27727992 0.73 CNR2 (0.49) ALDH1A1
SCHEMBL28136805 0.72 HDAC6 (0.49) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL17373675 0.72 SMN1; SMN2 (0.59) HDAC6HDAC3HDAC4HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945324-A Sulfur-based compound with anti-tumor activity and application thereof UNIV SHENYANG PHARMACEUTICAL 2015-09-30 CN claimed
CN-104945324-A Sulfur-based compound with anti-tumor activity and application thereof UNIV SHENYANG PHARMACEUTICAL 2015-09-30 CN disclosed