SCHEMBL28036356

SCHEMBL28036356

O=c1ccc2c(CC(F)(F)F)cccc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.40
DDO Q99489 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
AR P10275 7/20 0.38
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19326978 0.83 DAO (0.43) DAODDOCA12CA1CA3
SCHEMBL15108883 0.79 DAO (0.60) DAODDOCA12CA1CA3
SCHEMBL7425258 0.77 PDE3B (0.43) DAODDOCA12CA1CA3
SCHEMBL3787127 0.74 KIF11 (0.51) CA12CA1CA3CA4CA6
SCHEMBL30946245 0.74 KIF11 (0.51) CA12CA1CA3CA4CA6
SCHEMBL16338725 0.73 PDE3B (0.55) DAODDOCA12CA1CA3
SCHEMBL31557870 0.73 PDE3B (0.55) DAODDOCA12CA1CA3
SCHEMBL429173 0.73 NPC1 (0.45) DAODDOCA12CA1CA3
SCHEMBL1082903 0.71 DAO (0.53) DAODDOCA12CA1CA3
SCHEMBL3874061 0.71 KDM4E (0.60) DAODDOCA12CA1CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102453-A Benzimidazolone derivatives as bromodomain inhibitors GILEAD SCIENCES INC 2015-11-25 CN disclosed