SCHEMBL28039591

SCHEMBL28039591

FC(F)(F)Oc1cccc2c1NCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.44
OPRM1 P35372 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HTR2C P28335 3/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.35
GRIA1 P42261 3/20 0.34
CACNG8 Q8WXS5 3/20 0.34
CACNG2 Q9Y698 1/20 0.34
DDB1 Q16531 2/20 0.33
CRBN Q96SW2 2/20 0.33
PARP10 Q53GL7 2/20 0.33
PARP11 Q9NR21 2/20 0.33
PDPK1 O15530 1/20 0.33
PARP1 P09874 1/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33
CCR3 P51677 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10912135 0.90 SRC (0.56) SRCOPRM1KDM4EHTR2CHTR2B
SCHEMBL31238797 0.77 CES1 (0.40) SRCKDM4EHTR2CHTR2BHTR2A
SCHEMBL4795981 0.77 SRC (0.47) SRCPARP1
SCHEMBL25209388 0.77 CES1 (0.40) SRCKDM4EHTR2CHTR2BHTR2A
SCHEMBL21225396 0.75 SRC (0.39) SRCHTR2APARP10PARP11PARP1
SCHEMBL18355372 0.73 SRC (0.56) SRCPARP1KCNH2
SCHEMBL31158661 0.72 NOTUM (0.37) KDM4EHTR2CHTR2BHTR2AGRIA1
SCHEMBL12475573 0.72 NOTUM (0.37) KDM4EHTR2CHTR2BHTR2AGRIA1
SCHEMBL4718545 0.72 SRC (0.44) SRCHTR2CHTR2BPARP10PARP11
SCHEMBL27846115 0.72 SRC (0.44) SRCHTR2CPARP10PARP11PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073741-A Phthalazinones and isoquinolinones as rock inhibitors BRISTOL MYERS SQUIBB CO 2015-11-18 CN disclosed