SCHEMBL28039679

SCHEMBL28039679

COC(=O)c1ccc2c3ccccc3n(Cc3ccccc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC10 Q969S8 1/20 0.56
CYP19A1 P11511 1/20 0.55
S1PR3 Q99500 2/20 0.55
HDAC3 O15379 1/20 0.53
MAPT P10636 3/20 0.53
ALDH1A1 P00352 1/20 0.53
GAA P10253 1/20 0.53
PKM P14618 1/20 0.53
CNR2 P34972 1/20 0.53
THRB P10828 1/20 0.51
CFTR P13569 1/20 0.51
MAPK8 P45983 1/20 0.50
P2RX4 Q99571 1/20 0.50
F10 P00742 2/20 0.49
MAPK1 P28482 1/20 0.49
ATM Q13315 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13011553 0.90 P2RX4 (0.61) HDAC6HDAC1HDAC10S1PR3HDAC3
SCHEMBL13011224 0.90 CNR2 (0.55) HDAC6HDAC1HDAC10S1PR3HDAC3
SCHEMBL13011250 0.88 MAPT (0.53) HDAC6HDAC1MAPTALDH1A1THRB
SCHEMBL13011336 0.88 MAPT (0.51) HDAC6HDAC1HDAC10S1PR3HDAC3
SCHEMBL1002975 0.88 HDAC6 (0.67) HDAC6HDAC1HDAC10CYP19A1HDAC3
SCHEMBL13011169 0.87 CNR2 (0.58) HDAC6S1PR3HDAC3ALDH1A1CNR2
SCHEMBL13011342 0.86 HTT (0.52) HDAC6HDAC1HDAC10MAPTALDH1A1
SCHEMBL13011271 0.85 ROCK2 (0.51) HDAC6HDAC1HDAC10S1PR3HDAC3
SCHEMBL8388868 0.85 CYP19A1 (0.60) HDAC6HDAC1HDAC10CYP19A1HDAC3
SCHEMBL28039674 0.85 CYP19A1 (0.64) HDAC6HDAC1HDAC10CYP19A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008352-A Carbazole compounds useful as bromodomain inhibitors BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed