SCHEMBL28040054

SCHEMBL28040054

CC1(C)CNCCC1=O.O=COCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
HTR2C P28335 4/20 0.33
HTR2A P28223 2/20 0.33
MMP2 P08253 1/20 0.33
MMP13 P45452 1/20 0.33
HTR2B P41595 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
TACR1 P25103 1/20 0.33
TYK2 P29597 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HPGD P15428 1/20 0.32
PTPN1 P18031 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17956886 0.79 HTR2C (0.40) HTR2CHTR2AHTR2BTACR1SLC6A2
SCHEMBL28039720 0.77 ALDH1A1 (0.37) ALDH1A1
Piperazine SCHEMBL28083640 0.76 TACR1 (0.42) HTR2CHTR2AHTR2BTACR1SLC6A2
Azetidine SCHEMBL27976635 0.76 TSHR (0.41) ALDH1A1HTR2CTACR1SLC6A2SLC6A4
Piperazine SCHEMBL27484195 0.76 TACR1 (0.42) HTR2CHTR2AHTR2BTACR1SLC6A2
SCHEMBL27625376 0.76 CHRM2 (0.39) HTR2CHTR2AHTR2BTYK2
SCHEMBL28504837 0.75 HTR2C (0.36) ALDH1A1HTR2CMMP2MMP13HTR2B
Piperazine SCHEMBL28258210 0.75 TACR1 (0.41) HTR2CHTR2AHTR2BTACR1SLC6A2
SCHEMBL28826190 0.75 HTR2C (0.40) HTR2CHTR2AHTR2BTACR1SLC6A2
SCHEMBL28289813 0.74 TACR1 (0.43) ALDH1A1HTR2CTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105025899-A Having a2AHeterobicyclically substituted- [1 ] with antagonist properties MERCK SHARP & DOHME 2015-11-04 CN disclosed