SCHEMBL28040740

SCHEMBL28040740

CN(c1ccccc1CCBr)S(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
CLK2 P49760 1/20 0.41
AURKB Q96GD4 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
JAK2 O60674 2/20 0.40
PTK2 Q05397 2/20 0.40
JAK3 P52333 1/20 0.40
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
CDC42BPA Q5VT25 1/20 0.38
SRPK1 Q96SB4 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
MEN1 O00255 2/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
CYP19A1 P11511 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2634191 0.86 KMT2A (0.46) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL2634907 0.83 TAAR1 (0.44) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL16570034 0.83 KMT2A (0.44) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL10229066 0.82 KMT2A (0.49) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL30621311 0.79 KMT2A (0.46) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL16580719 0.79 KMT2A (0.46) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL646500 0.79 KMT2A (0.50) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL1291311 0.79 KMT2A (0.46) KMT2ACLK2AURKBCLK4JAK2
SCHEMBL646441 0.79 KMT2A (0.46) KMT2ACLK2AURKBCLK4JAK2
Hydrochloric Acid SCHEMBL30468480 0.77 KMT2A (0.45) KMT2ACLK2AURKBCLK4JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102459258-B Preparation and use of 1,2, 4-triazolo [1,5a ] pyridine derivatives CEPHALON, INC. (US) 2015-11-25 CN disclosed