SCHEMBL28041311

SCHEMBL28041311

COCC1CCCN1c1cccc(-c2cnc3cc(C(=O)O)ccc3n2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.49
HPGD P15428 6/20 0.42
ADORA2A P29274 4/20 0.42
ADORA1 P30542 4/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
LDHA P00338 1/20 0.41
LDHB P07195 1/20 0.41
P2RY12 Q9H244 1/20 0.40
IDH1 O75874 2/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28041187 0.89 SYK (0.47) SYKHPGDNPC1RAB9ALDHA
SCHEMBL27868874 0.85 HPGD (0.46) SYKHPGDNPC1RAB9ALDHA
SCHEMBL27868871 0.83 HPGD (0.45) HPGDNPC1RAB9ALDHALDHB
SCHEMBL1458828 0.77 HPGD (0.52) SYKHPGDADORA2AADORA1NPC1
SCHEMBL9949901 0.77 HPGD (0.52) SYKHPGDADORA2AADORA1NPC1
SCHEMBL27885415 0.77 HPGD (0.56) HPGDJAK2JAK3
SCHEMBL27868880 0.75 CHEK1 (0.52) HPGDNPC1RAB9AJAK2JAK3
SCHEMBL2277781 0.74 SYK (0.52) SYKJAK2JAK3
SCHEMBL27868895 0.74 NEK2 (0.41) HPGDADORA2ANPC1RAB9AJAK2
SCHEMBL27868873 0.73 ABCG2 (0.53) HPGDJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102656163-B Suppress the heterogeneous ring compound of PASK BIOENERGENIX (US) 2016-01-13 CN claimed
CN-102656163-B Suppress the heterogeneous ring compound of PASK BIOENERGENIX (US) 2016-01-13 CN disclosed