SCHEMBL28042019

SCHEMBL28042019

COC(=O)c1ccc(C(=O)O)n1NC(=S)NC(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
MAPT P10636 5/20 0.52
KMT2A Q03164 5/20 0.52
KDM4E B2RXH2 3/20 0.52
MEN1 O00255 3/20 0.52
ALOX12 P18054 2/20 0.52
HPGD P15428 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
EPHX1 P07099 4/20 0.47
GAA P10253 3/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
CCR6 P51684 1/20 0.44
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL520581 0.80 MAPT (0.49) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL519468 0.79 ALDH1A1 (0.52) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL17611061 0.77 ALDH1A1 (0.46) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL30020977 0.76 ALDH1A1 (0.46) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL522109 0.75 KMT2A (0.48) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL18689666 0.75 ALDH1A1 (0.48) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL29943719 0.72 EPHX1 (0.50) ALDH1A1KMT2AKDM4EMEN1ALOX12
SCHEMBL19222024 0.72 ALDH1A1 (0.50) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL31398632 0.70 ALDH1A1 (0.77) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL24747452 0.68 ALDH1A1 (0.60) ALDH1A1MAPTKMT2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105130992-A Nitrogen-containing heterocyclic compound having kinase inhibiting activity, preparation method and application UNIV SOOCHOW 2015-12-09 CN disclosed