SCHEMBL28042449

SCHEMBL28042449

Br[Mg]Br.Fc1cccc(-c2cc[c]cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.50
ESR2 Q92731 1/20 0.50
CYP17A1 P05093 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTPN1 P18031 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
IDO1 P14902 2/20 0.36
NOTUM Q6P988 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
KDM4E B2RXH2 3/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316987 0.92 TAAR1 (0.57) TAAR1ESR2CYP17A1CYP3A4CYP11B1
SCHEMBL28311259 0.90 TAAR1 (0.55) TAAR1ESR2CYP17A1CYP3A4CYP11B1
SCHEMBL28042450 0.77 BCL2L1 (0.37) CYP11B1CYP11B2PTPN1
SCHEMBL19471215 0.77 ALDH1A1 (0.47) TAAR1ESR2CYP3A4NOTUMKDM4E
SCHEMBL11973522 0.76 MEN1 (0.48) TAAR1ESR2CYP3A4NISCHHSD17B1
SCHEMBL198702 0.76 TAAR1 (0.68) TAAR1ESR2CYP17A1CYP3A4CYP11B1
Biphenyl SCHEMBL25183774 0.74 TAAR1 (0.67) TAAR1ESR2CYP17A1CYP3A4CYP11B1
SCHEMBL29451178 0.74 TAAR1 (0.67) TAAR1ESR2CYP17A1CYP3A4CYP11B1
SCHEMBL200605 0.74 TAAR1 (0.67) TAAR1ESR2CYP17A1CYP3A4CYP11B1
SCHEMBL16605626 0.73 TAAR1 (0.65) TAAR1ESR2CYP17A1CYP3A4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105101967-A Benzazepines as serotonin 5-ht2c receptor ligands and uses thereof ABT HOLDING CO 2015-11-25 CN disclosed